Mallamo, John P.: search on Z-Library

The world's largest scientific articles store. 70,000,000+ articles for free.

1

Antiandrogenic steroidal sulfonylpyrazoles

Christiansen, Robert G., Bell, Malcolm R., D'Ambra, Thomas E., Mallamo, John P., Herrmann, John L., Ackerman, James H., Opalka, Chester J., Kullnig, Rudolph K., Winneker, Richard C.

Journal:

Journal of Medicinal Chemistry

Year:

1990

Language:

english

File:

PDF, 1.77 MB

english, 1990

2

Synthesis and Mixed Lineage Kinase Activity of Pyrrolocarbazole and Isoindolone Analogs of (+)K-252a

Hudkins, Robert L., Johnson, Neil W., Angeles, Thelma S., Gessner, George W., Mallamo, John P.

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 156 KB

english, 2007

3

Nonpeptidic inhibitors of recombinant human calpain I

Sankar Chatterjee, Shobha Senadhi, Donna Bozyczko-Coyne, Robert Siman, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 182 KB

english, 1997

4

Antiandrogenic steroidal sulfonyl heterocycles. Utility of electrostatic complementarity in defining bioisosteric sulfonyl heterocycles

Mallamo, John P., Pilling, Garry M., Wetzel, Joseph R., Kowalczyk, Paul J., Bell, Malcolm R., Kullnig, Rudolph K., Batzold, Frederick H., Juniewicz, Paul E., Winneker, Richard C., Luss, Henry R.

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 2.07 MB

english, 1992

5

Syntheses of C12,N13 Heterocyclic Bridged Fused Indenopyrrolocarbazoles.

Ted L. Underiner, John P. Mallamo, Jasbir Singh

Journal:

Year:

2002

File:

PDF, 30 KB

2002

6

Potent α-ketocarbonyl and boronic ester derived inhibitors of proteasome

Mohamed Iqbal, Sankar Chatterjee, James C. Kauer, John P. Mallamo, Patricia A. Messina, Alyssa Reiboldt, Robert Siman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 160 KB

english, 1996

7

Exploration of the importance of the P2-P3 -NHCO-Moiety in a potent di- or tripeptide inhibitor of calpain i: insights into the development of nonpeptidic inhibitors of calpain I

Sankar Chatterjee, Mohamed Iqbal, Satish Mallya, Shobha E. Senadhi, Teresa M. O’Kane, Beth Ann McKenna, Donna Bozyczko-Coyne, James C. Kauer, Robert Siman, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 257 KB

english, 1998

8

Novel NMDA Antagonists: Replacement of the Pyridinium Ring of 6,11-Ethanobenzo[b]quinolizinium Cations with Heteroisoquinolinium Cations

Kumar, Virendra, Carabateas, Phil M., Dority, John A., Earley, William G., Mallamo, John P., Subramanyam, Chakrapani, Aimone, Lisa D., Ault, Brian, Hudkins, Diane L. DeHaven, Miller, Matthew S.

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 615 KB

english, 1995

9

Xanthene derived potent nonpeptidic inhibitors of recombinant human calpain I

Sankar Chatterjee, Mohamed Iqbal, James C. Kauer, John P. Mallamo, Shobha Senadhi, Satish Mallya, Donna Bozyczko-Coyne, Robert Siman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 230 KB

english, 1996

10

Preclinical evaluation of acylhydrazone SB-AF-1002 as a novel broad-spectrum antifungal agent

Lazzarini, Cristina, Haranahalli, Krupanandan, McCarthy, J. Brian, Mallamo, John, Ojima, Iwao, Del Poeta, Maurizio

Journal:

Antimicrobial Agents and Chemotherapy

Year:

2020

File:

PDF, 2.58 MB

2020

11

TrkA kinase inhibitors from a library of modified and isosteric Staurosporine aglycone

Rabindranath Tripathy, Thelma S. Angeles, Shi X. Yang, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 195 KB

english, 2008

12

1,2-Benzothiazine 1,1-dioxide α-ketoamide analogues as potent calpain I inhibitors

Ron Bihovsky, Ming Tao, John P. Mallamo, Gregory J. Wells

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2004

Language:

english

File:

PDF, 169 KB

english, 2004

13

Knowledge-Based, Central Nervous System (CNS) Lead Selection and Lead Optimization for CNS Drug Discovery

Ghose, Arup K., Herbertz, Torsten, Hudkins, Robert L., Dorsey, Bruce D., Mallamo, John P.

Journal:

ACS Chemical Neuroscience

Year:

2012

Language:

english

File:

PDF, 3.74 MB

english, 2012

14

Discovery of 6,11-Ethano-12,12-diaryl-6,11-dihydrobenzo[b]quinolizinium Cations, a Novel Class of N-Methyl-D-aspartate Antagonists

Subramanyam, Chakrapani, Mallamo, John P., Dority, John A., Earley, William G., Kumar, Virendra, Aimone, Lisa D., Ault, Brian, Miller, Matthew S., Luttinger, Daniel A., DeHaven-Hudkins, Diane L.

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 824 KB

english, 1995

15

Syntheses of C12,N13 Heterocyclic Bridged Fused Indenopyrrolocarbazoles

Underiner, Ted L., Mallamo, John P., Singh, Jasbir

Journal:

Journal of Organic Chemistry

Year:

2002

Language:

english

File:

PDF, 122 KB

english, 2002

16

A convenient synthesis of 3-substituted pipecolic acid methyl esters

Chakrapani Subramanyam, Sankar Chattarjee, John P Mallamo

Journal:

Tetrahedron Letters

Year:

1996

Language:

english

File:

PDF, 157 KB

english, 1996

17

Regiocontrolled Syntheses of Benzo[b]quinolizinium and Heteroisoquinolinium Cations

G. Earley, William, A. Dority Jr., John, Kumar, Virendra, P. Mallamo, John

Journal:

Year:

1995

Language:

english

File:

PDF, 159 KB

english, 1995

18

1,2-Benzothiazine 1,1-Dioxide α-Ketoamide Analogues as Potent Calpain I Inhibitors.

Ron Bihovsky, Ming Tao, John P. Mallamo, Gregory J. Wells

Journal:

Year:

2004

File:

PDF, 90 KB

2004

19

Synthesis and Evaluation of 6,11-Ethanohexahydrobenzo[b]quinolizidines: A New Class of Noncompetitive N-Methyl-D-aspartate Antagonists

Subramanyam, Chakrapani, Mallamo, John P., Pilling, Gary M., Earley, William G., Carabateas, Philip M., Wetzel, Joseph R., DeHaven-Hudkins, Diane, Allen, Timothy, Kullnig, Rudolph K.

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 1.25 MB

english, 1995

20

Synthesis and structure-activity studies of some disubstituted phenylisoxazoles against human picornavirus

Diana, Guy D., Cutcliffe, David, Oglesby, Richard C., Otto, Michael J., Mallamo, John P., Akullian, Vahan, McKinlay, Mark A.

Journal:

Journal of Medicinal Chemistry

Year:

1989

Language:

english

File:

PDF, 672 KB

english, 1989

21

[Annual Reports in Medicinal Chemistry] Volume 24 || Chapter 21. New Horizons in the Treatment of Proliferative Prostatic Disease

Mallamo, John P.

Year:

1989

Language:

english

File:

PDF, 832 KB

english, 1989

22

The future of antifungal drug therapy: novel compounds and targets

Fernandes, Caroline Mota, Dasilva, Deveney, Haranahalli, Krupanandan, McCarthy, J. Brian, Mallamo, John, Ojima, Iwao, Del Poeta, Maurizio

Journal:

Antimicrobial Agents and Chemotherapy

Year:

2020

File:

PDF, 1.59 MB

2020

23

Calpain inhibitors based on the quiescent affinity label concept: high rates of calpain inactivation with leaving groups derived from N-hydroxy peptide coupling reagents

Rabindranath Tripathy, Mark A. Ator, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 143 KB

english, 2000

24

Antirhinoviral activity of heterocyclic analogs of Win 54954

Bailey, Thomas R., Diana, Guy D., Kowalczyk, Paul J., Akullian, Vahan, Eissenstat, Michael A., Cutcliffe, David, Mallamo, John P., Carabateas, Philip M., Pevear, Daniel C.

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 608 KB

english, 1992

25

Appendix: Correlation of Pocket Size and Shape with Antiviral Activity

Guy Diana, John P. Mallamo

Journal:

Journal of Molecular Biology

Year:

1993

File:

PDF, 93 KB

1993

26

Tandem michael-michael-ring closure (mimirc) reactions: One-pot steroid total synthesis-(±)-9,11-dehydroestrones

Gary H. Posner, John P. Mallamo, Alison Y. Black

Journal:

Year:

1981

Language:

english

File:

PDF, 614 KB

english, 1981

27

Knowledge Based Prediction of Ligand Binding Modes and Rational Inhibitor Design for Kinase Drug Discovery

Ghose, Arup K., Herbertz, Torsten, Pippin, Douglas A., Salvino, Joseph M., Mallamo, John P.

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 1.44 MB

english, 2008

28

High asymmetric induction during organometallic .beta.-addition to .alpha.,.beta.-ethylenic sulfoxides. Synthesis of optically active .beta.-alkylcarboxylic acids, .beta.-substituted cyclopentanones, and steroidal 11-oxoequilenin methyl ether

Posner, Gary H., Mallamo, John P., Miura, Kyo

Journal:

Journal of the American Chemical Society

Year:

1981

Language:

english

File:

PDF, 377 KB

english, 1981

29

P2-achiral, P'-extended α-ketoamide inhibitors of calpain I

Sankar Chatterjee, Derek Dunn, Ming Tao, Gregory Wells, Zi-Qiang Gu, Ron Bihovsky, Mark A. Ator, Robert Siman, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 209 KB

english, 1999

30

Structure-activity studies of 5-[[4-(4,5-dihydro-2-oxazolyl)phenoxy]alkyl]-3-methylisoxazoles: inhibitors of picornavirus uncoating

Diana, Guy D., Oglesby, Richard C., Akullian, Vahan, Carabateas, Philip M., Cutcliffe, David, Mallamo, John P., Otto, Michael J., McKinlay, Mark A., Maliski, Edward G., Michalec, Stephen J.

Journal:

Journal of Medicinal Chemistry

Year:

1987

Language:

english

File:

PDF, 761 KB

english, 1987

31

An Evaluation of the Antirhinoviral Activity of Acylfuran Replacements for 3-Methylisoxazoles. Are 2-Acetylfurans Bioisosteres for 3-Methylisoxazoles? [Erratum to document cited in CA122:31229]

Bailey, Thomas R., Diana, Guy D., Mallamo, John P., Vescio, Niranjan, Draper, Tandy L., Carabateas, Philip M., Long, Melody A., Giranda, Vincent L., Dutko, Frank J., Pevear, Daniel C.

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 56 KB

english, 1995

32

Novel Peptidyl Phosphorus Derivatives as Inhibitors of Human Calpain I

Tao, Ming, Bihovsky, Ron, Wells, Gregory J., Mallamo, John P.

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 86 KB

english, 1998

33

Knowledge-based chemoinformatic approaches to drug discovery

Arup K. Ghose, Torsten Herbertz, Joseph M. Salvino, John P. Mallamo

Journal:

Drug Discovery Today

Year:

2006

Language:

english

File:

PDF, 728 KB

english, 2006

34

ChemInform Abstract: Calpain Inhibitors Based on the Quiescent Affinity Label Concept: High Rates of Calpain Inactivation with Leaving Groups Derived from N-Hydroxy Peptide Coupling Reagents.

Rabindranath Tripathy, Mark A. Ator, John P. Mallamo

Journal:

Year:

2001

File:

PDF, 30 KB

2001

35

Potent fluoromethyl ketone inhibitors of recombinant human calpain I

Sankar Chatterjee, Kurt Josef, Gregory Wells, Mohamed Iqbal, Ron Bihovsky, John P. Mallamo, Mark A. Ator, Donna Bozyczko-Coyne, Satish Mallya, Shobha Senadhi, Robert Siman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 230 KB

english, 1996

36

Asymmetric induction during organometallic conjugate addition to enantiomerically pure 2-(arylsulfinyl)-2-cyclopentenones

Posner, Gary H., Mallamo, John P., Hulce, Martin, Frye, Leah L.

Journal:

Journal of the American Chemical Society

Year:

1982

Language:

english

File:

PDF, 884 KB

english, 1982

37

Generation and reactions of 1-(arylsulfinyl)alkenyllithium reagents. Terminal allenes from 2-alkenyl aryl sulfoxides.

Gary H. Posner, Ping-Wah Tang, John P. Mallamo

Journal:

Tetrahedron Letters

Year:

1978

Language:

english

File:

PDF, 212 KB

english, 1978

38

Identification, Synthesis, and Characterization of a Unique Class of N-Methyl-D-aspartate Antagonists. The 6,11-Ethanobenzo[b]quinolizinium Cation

Mallamo, John P., Earley, William G., Kumar, Virendra, Subramanyam, Chakrapani, Dority, John A. Jr., Miller, Matthew S., DeHaven-Hudkins, Diane L., Ault, Brian, Herrmann, John L.

Journal:

Journal of Medicinal Chemistry

Year:

1994

Language:

english

File:

PDF, 2.62 MB

english, 1994

39

1,2,3-Thiadiazole substituted pyrazolones as potent KDR/VEGFR-2 kinase inhibitors

Rabindranath Tripathy, Arup Ghose, Jasbir Singh, Edward R. Bacon, Thelma S. Angeles, Shi X. Yang, Mark S. Albom, Lisa D. Aimone, Joseph L. Herman, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 248 KB

english, 2007

40

A simple synthetic protocol for the protection of amides, lactams, ureas, and carbamates

Dandu R Reddy, Mohamed A Iqbal, Robert L Hudkins, Patricia A Messina-McLaughlin, John P Mallamo

Journal:

Tetrahedron Letters

Year:

2002

Language:

english

File:

PDF, 179 KB

english, 2002

41

Improved resolution of (±)-trans-2'-hydroxy-5,9-dimethyl-6,7-benzomorphans

Joseph R. Wetzel, John D. Grego, John P. Mallamo

Journal:

Year:

1992

Language:

english

File:

PDF, 331 KB

english, 1992

42

A Simple Synthetic Protocol for the Protection of Amides, Lactams, Ureas, and Carbamates.

Dandu R. Reddy, Mohamed A. Iqbal, Robert L. Hudkins, Patricia A. Messina-McLaughlin, John P. Mallamo

Journal:

Year:

2003

File:

PDF, 119 KB

2003

43

Construction of a kinase inhibitor library via parallel synthesis

Rabindranath Tripathy, Keith S Learn, Dandu R Reddy, Mohamed Iqbal, Jasbir Singh, John P Mallamo

Journal:

Tetrahedron Letters

Year:

2002

Language:

english

File:

PDF, 147 KB

english, 2002

44

Synthesis and binding affinity of 2,3,3a,4,9,9a-hexahydro-9,4-(iminomethano)-1H-benz[f]indenes. Ligands for the PCP site of the NMDA receptor

Michael Reuman, John P. Mallamo, Diane L. DeHaven-Hudkins

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 238 KB

english, 1995

45

Synthesis of deuterium-labeled 5α-androstane-3α,17β-diol and its 17β-glucuronide

Chung Bong-Chul, John P. Mallamo, Paul E. Juniewicz, Cedric H.L. Shackleton

Journal:

Year:

1992

Language:

english

File:

PDF, 711 KB

english, 1992

46

Complete asymmetric induction in synthesis of enantiomerically pure steroid intermediates of natural configuration

Posner, Gary H., Hulce, Martin, Mallamo, John P., Drexler, Steven A., Clardy, Jon

Journal:

Journal of Organic Chemistry

Year:

1981

Language:

english

File:

PDF, 388 KB

english, 1981

47

Antipicornavirus activity of tetrazole analogs related to disoxaril

Diana, Guy D., Cutcliffe, David, Volkots, Deborah L., Mallamo, John P., Bailey, Thomas R., Vescio, Niranjan, Oglesby, Richard C., Nitz, Theodore J., Wetzel, Joseph

Journal:

Journal of Medicinal Chemistry

Year:

1993

Language:

english

File:

PDF, 2.11 MB

english, 1993

48

SAR Studies on Aromatic Acylhydrazone-Based Inhibitors of Fungal Sphingolipid Synthesis as Next-Generation Antifungal Agents

Haranahalli, Krupanandan, Lazzarini, Cristina, Sun, Yi, Zambito, Julia, Pathiranage, Senuri, McCarthy, John Brian, Mallamo, John P., Del Poeta, Maurizio, Ojima, Iwao

Journal:

Journal of Medicinal Chemistry

Year:

2019

Language:

english

File:

PDF, 1.11 MB

english, 2019

49

Prodrug esters of the indolocarbazole CEP-751 (KT-6587)

Robert L. Hudkins, Mohamed Iqbal, Chung-Ho Park, Joel Goldstein, Joseph L. Herman, Efraim Shek, Chikara Murakata, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 212 KB

english, 1998

50

Novel Benzo[b]quinolizinium Cations as Uncompetitive N-Methyl-D-aspartic Acid (NMDA) Antagonists: The Relationship between log D and Agonist Independent (Closed) NMDA Channel Block

Earley, William G., Kumar, Virendra, Mallamo, John P., Subramanyam, Chakrapani, Dority, John A., Miller, Matthew S., DeHaven-Hudkins, Diane L., Aimone, Lisa D., Kelly, Michael D., Ault, Brian

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 1.00 MB

english, 1995

To build up a library is to create a life. It’s never just a random collection of books.

— Carlos María Domínguez

Official channel

Z-Library Desktop Launcher

Z-Library Since 2009 support@1delivery.pm

EnglishРусскийEspañolItalianoελληνικάاللغة العربيةBahasa IndonesiaBahasa Malaysiaहिन्दीDeutschFrançaisPortuguêsУкраїнськаPolski中文繁體中文日本語Tiếng ViệtAzərbaycan DiliՀայոց լեզուภาษาไทยTürk Diliქართველიবাংলাپښتوతెలుగుاردو한국어SrpskiБългарски